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Design ,Synthesis, Insilco Study and Biological Evaluation of New Coumarin-Oxadiazole Derivatives as Potent Histone Deacetylase Inhibitors

Abstract
A new series of HDAC inhibitors were designed, synthesized, bearing acyl semicarbazide, hydrazide and hydrazide derivatives as ZBGs, alkyl thio oxadiazole as the linker group and coumarin as the cap group .These derivatives were evaluated for their HDACs inhibitory activities against MDA-MB-231 (a human breast cancer cell line) and HepG2 (a human hepatocellular carcinoma cell line), most of them h...
Keywords
Coumarin
Histone deacetylase
Oxadiazole
Chemistry
Histone deacetylase inhibitor
Pharmacology
Combinatorial chemistry
Histone
Biochemistry
Medicine
Organic chemistry
DNA



Design ,Synthesis, Insilco Study and Biological Evaluation of New Coumarin-Oxadiazole Derivatives as Potent Histone Deacetylase Inhibitors

Design ,Synthesis, Insilco Study and Biological Evaluation of New Coumarin-Oxadiazole Derivatives as Potent Histone Deacetylase Inhibitors

Abstract
A new series of HDAC inhibitors were designed, synthesized, bearing acyl semicarbazide, hydrazide and hydrazide derivatives as ZBGs, alkyl thio oxadiazole as the linker group and coumarin as the cap group .These derivatives were evaluated for their HDACs inhibitory activities against MDA-MB-231 (a human breast cancer cell line) and HepG2 (a human hepatocellular carcinoma cell line), most of them h...
Keywords
Coumarin
Histone deacetylase
Oxadiazole
Chemistry
Histone deacetylase inhibitor
Pharmacology
Combinatorial chemistry
Histone
Biochemistry
Medicine
Organic chemistry
DNA